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Fungal biotransformation of 1,3-oxathiolanes

 

作者: Herbert L. Holland,   Benito Munoz,  

 

期刊: Canadian Journal of Chemistry  (NRC Available online 1988)
卷期: Volume 66, issue 9  

页码: 2299-2303

 

ISSN:0008-4042

 

年代: 1988

 

DOI:10.1139/v88-364

 

出版商: NRC Research Press

 

数据来源: NRC

 

摘要:

A series of 2,2-disubstituted 1,3-oxathiolanes has been incubated with fungi known to be capable of efficient asymmetric oxidation of sulfides to sulfoxides. In three cases (2-phenyl-1,3-oxathiolane, 2-methyl-2-phenyl-1,3-oxathiolane, and 2-tert-butyl-2-phenyl-1,3-oxathiolane), sulfoxidation occurred to give a single diastereomer of sulfoxide, whose relative stereochemistry has been assigned by1H nuclear magnetic resonance analysis. The sulfoxides were obtained as racemates or had low enantiomeric enrichment. In some cases ketones, assumed to be formed by spontaneous hydrolysis of oxathiolane sulfoxides, were obtained, together with their reduction products, secondary alcohols.

 

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